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Horta P, Kuş N, Henriques MSofia C, et al. Quinolone-Hydroxyquinoline Tautomerism in Quinolone 3-Esters. Preserving the 4-Oxoquinoline Structure To Retain Antimalarial Activity. J Org Chem. 2015;80(24):12244-57. doi:10.1021/acs.joc.5b02169
R
W. Hong D, Gibbons PD, Leung SC, et al. Rational Design, Synthesis, and Biological Evaluation of Heterocyclic Quinolones Targeting the Respiratory Chain of Mycobacterium tuberculosis. Journal of Medicinal Chemistry. 2017;60(9):3703 - 3726. doi:10.1021/acs.jmedchem.6b01718